Medicines
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Generic: CGP 54626
CGP 54626 is a potent and selective antagonist of the GABA<sub>B</sub> receptor. It is a research tool primarily used in scientific studies to investigate the role and function of GABA<sub>B</sub> receptors in various physiological and pathological processes.
Used in research to block GABA<sub>B</sub> receptors and study their function.
Outcome:
Reduced efficacy of baclofen
Mechanism:
Competitive antagonism at GABA<sub>B</sub> receptors.
Outcome:
Potential decreased seizure control.
Mechanism:
Interference with GABAergic modulation.
Outcome:
Potential minor interaction due to opposing effects on CNS.
Mechanism:
Stimulatory vs. inhibitory effects.
No significant innovation is forecast for this primarily research-focused compound.
Due to its limited clinical use, no regulatory predictions can be made.
GABA<sub>B</sub> Receptor Antagonist
Pyridine Derivative